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1

Synthesis of 5- and 6-substituted 2-(4-dimethylaminophenyl)-1,3-benzoxazoles and their in vitro and in vivo evaluation as imaging agents for amyloid plaque

Sven H. Hausner, David Alagille, Andrei O. Koren, Louis Amici, Julie K. Staley, Kelly P. Cosgrove, Ronald M. Baldwin, Gilles D. Tamagnan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 152 KB

english, 2009

2

Microwave-induced nucleophilic [18F]fluorination on aromatic rings: Synthesis and effect of halogen on [18F]fluoride substitution of meta-halo (F, Cl, Br, I)-benzonitrile derivatives

Ning Guo, David Alagille, Gilles Tamagnan, Ronald R. Price, Ronald M. Baldwin

Journal:

Applied Radiation and Isotopes

Year:

2008

Language:

english

File:

PDF, 283 KB

english, 2008

3

GABAA-benzodiazepine receptor availability in smokers and nonsmokers: Relationship to subsyndromal anxiety and depression

Irina Esterlis, Kelly P. Cosgrove, Jeffery C. Batis, Frederic Bois, Tracy A. Kloczynski, Stephanie M. Stiklus, Edward Perry, Gilles D. Tamagnan, John P. Seibyl, Robert Makuch, Suchitra Krishnan-Sarin,

Journal:

Year:

2009

Language:

english

File:

PDF, 178 KB

english, 2009

4

A novel 18 F-labelled high affinity agent for PET imaging of the translocator protein

Blair, Adele, Zmuda, Filip, Malviya, Gaurav, Tavares, Adriana A. S., Tamagnan, Gilles D., Chalmers, Anthony J., Dewar, Deborah, Pimlott, Sally L., Sutherland, Andrew

Journal:

Chemical Science

Year:

2015

Language:

english

File:

PDF, 2.90 MB

english, 2015

5

Identification and in vivo evaluation of a fluorine-18 rolipram analogue, [ 18 F]MNI-617, as a radioligand for PDE4 imaging in mammalian brain

Thomae, David, Morley, Thomas J., Lee, Hsiaoju S., Barret, Olivier, Constantinescu, Cristian, Papin, Caroline, Baldwin, Ronald M., Tamagnan, Gilles D., Alagille, David

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2016

Language:

english

File:

PDF, 1.69 MB

english, 2016

6

Comparison between [ 18 F]fluorination and [ 18 F]fluoroethylation reactions for the synthesis of the PDE10A PET radiotracer [ 18 F]MNI-659

Mori, Wakana, Takei, Makoto, Furutsuka, Kenji, Fujinaga, Masayuki, Kumata, Katsushi, Muto, Masatoshi, Ohkubo, Takayuki, Hashimoto, Hiroki, Tamagnan, Gilles, Higuchi, Makoto, Kawamura, Kazunori, Zhang,

Journal:

Nuclear Medicine and Biology

Year:

2017

Language:

english

File:

PDF, 654 KB

english, 2017

7

18F-F13640 preclinical evaluation in rodent, cat and primate as a 5-HT1A receptor agonist for PET neuroimaging

Vidal, Benjamin, Fieux, Sylvain, Colom, Matthieu, Billard, Thierry, Bouillot, Caroline, Barret, Olivier, Constantinescu, Cristian, Tamagnan, Gilles, Newman-Tancredi, Adrian, Zimmer, Luc

Journal:

Brain Structure and Function (Anatomy and Embryology 1891-2006)

Year:

2018

Language:

english

File:

PDF, 2.36 MB

english, 2018

8

Intrastriatal alpha-synuclein fibrils in monkeys: spreading, imaging and neuropathological changes

Chu, Yaping, Muller, Scott, Tavares, Adriana, Barret, Olivier, Alagille, David, Seibyl, John, Tamagnan, Gilles, Marek, Ken, Luk, Kelvin C, Trojanowski, John Q, Lee, Virginia M Y, Kordower, Jeffrey H

Journal:

Year:

2019

Language:

english

File:

PDF, 434 KB

english, 2019

9

Biomarkers for Parkison's disease: Tools to assess Parkinson's disease onset and progression

Kenneth Marek, Danna Jennings, Gilles Tamagnan, John Seibyl

Journal:

Annals of Neurology

Year:

2008

Language:

english

File:

PDF, 130 KB

english, 2008

10

ChemInform Abstract: Synthesis and Monoamine Transporter Affinity of 2β-Carbomethoxy-3β-(2′′-, 3′′-, or 4′′-substituted) Biphenyltropanes.

Gilles Tamagnan, Ronald M. Baldwin, Nora S. Kula, Ross J. Baldessarini, Robert B. Innis

Journal:

Year:

2000

File:

PDF, 35 KB

2000

11

Synthesis and Monoamine Transporter Affinity of 3′-Analogues of 2-β-Carbomethoxy-3-β-(4′-iodophenyl)tropane (β-CIT).

Frederic Bois, Ronald M. Baldwin, Nora S. Kula, Ross J. Baldessarini, Robert B. Innis, Gilles Tamagnan

Journal:

Year:

2004

File:

PDF, 131 KB

2004

12

Total Synthesis of the Marine Cytotoxic Caulibugulones A—D.

David Alagille, Ronald M. Baldwin, Gilles D. Tamagnan

Journal:

Year:

2004

File:

PDF, 10 KB

2004

13

One-Step Synthesis of 2-Arylbenzothiazole (“BTA”) and -benzoxazole Precursors for in vivo Imaging of β-Amyloid Plaques.

David Alagille, Ronald M. Baldwin, Gilles D. Tamagnan

Journal:

Year:

2005

File:

PDF, 21 KB

2005

14

Functionalization at Position 3 of the Phenyl Ring of the Potent mGluR5 Noncompetitive Antagonists MPEP.

David Alagille, Ronald M. Baldwin, Bryan L. Roth, Jarda T. Wroblewski, Ewa Grajkowska, Gilles D. Tamagnan

Journal:

Year:

2005

File:

PDF, 20 KB

2005

15

Synthesis and Monoamine Transporter Affinity of New 2β-Carbomethoxy-3β-[4-(substituted thiophenyl)]phenyltropanes: Discovery of a Selective SERT Antagonist with Picomolar Potency.

Gilles Tamagnan, David Alagille, Xing Fu, Nora S. Kula, Ross J. Baldessarini, Robert B. Innis, Ronald M. Baldwin

Journal:

Year:

2005

File:

PDF, 25 KB

2005

16

Asymmetric Synthesis of (+)-(S,S)-Reboxetine via a New (S)-2-(Hydroxymethyl)morpholine Preparation.

Eric Brenner, Ronald M. Baldwin, Gilles Tamagnan

Journal:

Year:

2005

File:

PDF, 24 KB

2005

17

ChemInform Abstract: 2-Arylimidazo[2,1-b]benzothiazoles: A New Family of Amyloid Binding Agents with Potential for PET and SPECT Imaging of Alzheimer′s Brain.

David Alagille, Herve DaCosta, Ronald M. Baldwin, Gilles D. Tamagnan

Journal:

Year:

2011

File:

PDF, 25 KB

2011

18

Radiosynthesis of 3-(3-[18F]fluoropropoxy)-4-(benzyloxy)-N-[(1-dimethylaminocyclopentyl)methyl]-5-methoxybenzamide, a potential PET radiotracer for the glycine transporter GlyT-2

Haibin Tian, Rebecca Vogel, Louis Amici, Gilles Tamagnan, Ronald M. Baldwin

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2006

Language:

english

File:

PDF, 180 KB

english, 2006

19

6-[123I]Iodo-2-[[4-(2-methoxyphenyl) piperazin-1-yl]methyl]imidazo[1,2-a]pyridine as potential SPECT agent for imaging dopamine D4 receptor: synthesis and in vivo evaluation in a nonhuman primate

David Alagille, Andrei O. Koren, Greg Kudej, Julie Staley, Kelly Cosgrove, John Seibyl, Gilles D. Tamagnan

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2008

Language:

english

File:

PDF, 129 KB

english, 2008

20

An efficient synthesis of m-hydroxycocaine and m-hydroxybenzoylecgonine, two metabolites of cocaine

Gilles Tamagnan, Yigong Gao, Venkatesalu Bakthavachalam, William L. White, John L. Neumeyer

Journal:

Tetrahedron Letters

Year:

1995

Language:

english

File:

PDF, 174 KB

english, 1995

21

Synthesis of β-CIT-BAT, a potential technetium-99m imaging ligand for dopamine transporter

Gilles Tamagnan, Yigong Gao, Ronald M. Baldwin, Sami S. Zoghbi, John L. Neumeyer

Journal:

Tetrahedron Letters

Year:

1996

Language:

english

File:

PDF, 171 KB

english, 1996

22

Synthesis and receptor assay of aromatic–ethynyl–aromatic derivatives with potent mGluR5 antagonist activity

David Alagille, Ronald M. Baldwin, Bryan L. Roth, Jarda T. Wroblewski, Ewa Grajkowska, Gilles D. Tamagnan

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 380 KB

english, 2005

23

Synthesis and receptor binding studies of halogenated N,N-dialkylel-(2-phenyl-1H-indol-3-yl)glyoxylamides to visualize peripheral benzodiazepine receptors with SPECT or PET

Idriss Bennacef, Colin N. Haile, Anne Schmidt, Andrei O. Koren, John P. Seibyl, Julie K. Staley, Frederic Bois, Ronald M. Baldwin, Gilles Tamagnan

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 219 KB

english, 2006

24

Synthesis and affinity of a possible byproduct of electrophilic radiolabeling of [123I]IBZM

Ronald M Baldwin, Xing Fu, Nora S Kula, Ross J Baldessarini, Louis Amici, Robert B Innis, Gilles D Tamagnan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 135 KB

english, 2003

25

Synthesis and monoamine transporter affinity of 3′-analogs of 2-β-carbomethoxy-3-β-(4′-iodophenyl)tropane (β-CIT)

Frederic Bois, Ronald M Baldwin, Nora S Kula, Ross J Baldessarini, Robert B Innis, Gilles Tamagnan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2004

Language:

english

File:

PDF, 262 KB

english, 2004

26

Synthesis and monoamine transporter affinity of new 2β-carbomethoxy-3β-[4-(substituted thiophenyl)]phenyltropanes: discovery of a selective SERT antagonist with picomolar potency

Gilles Tamagnan, David Alagille, Xing Fu, Nora S. Kula, Ross J. Baldessarini, Robert B. Innis, Ronald M. Baldwin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 102 KB

english, 2005

27

Functionalization at position 3 of the phenyl ring of the potent mGluR5 noncompetitive antagonists MPEP

David Alagille, Ronald M. Baldwin, Bryan L. Roth, Jarda T. Wroblewski, Ewa Grajkowska, Gilles D. Tamagnan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 137 KB

english, 2005

28

Synthesis and monoamine transporter affinity of new 2β-carbomethoxy-3β-[aryl or heteroaryl]phenyltropanes

Gilles Tamagnan, David Alagille, Xing Fu, Nora S. Kula, Ross J. Baldessarini, Robert B. Innis, Ronald M. Baldwin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 138 KB

english, 2006

29

Synthesis and monoamine transporter affinity of 2β-carbomethoxy-3β-(4′-p-substituted phenyl)-piperidine analogs of cocaine

Frederic Bois, Ronald M. Baldwin, Nora S. Kula, Ross J. Baldessarini, M. Al Tikriti, Robert B. Innis, Gilles D. Tamagnan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 126 KB

english, 2006

30

Development of SPECT imaging agents for the norepinephrine transporters: [123I]INER

Gilles D. Tamagnan, Eric Brenner, David Alagille, Julie K. Staley, Colin Haile, Andrei Koren, Michelle Early, Ronald M. Baldwin, Frank I. Tarazi, Ross J. Baldessarini, Nachwa Jarkas, Mark M. Goodman,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 160 KB

english, 2007

31

2-Arylimidazo[2,1-b]benzothiazoles: A new family of amyloid binding agents with potential for PET and SPECT imaging of Alzheimer’s brain

David Alagille, Herve DaCosta, Ronald M. Baldwin, Gilles D. Tamagnan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 303 KB

english, 2011

32

Potent mGluR5 antagonists: Pyridyl and thiazolyl-ethynyl-3,5-disubstituted-phenyl series

David Alagille, Herve DaCosta, Yelin Chen, Kamondanai Hemstapat, Alice Rodriguez, Ronald M. Baldwin, Jeffrey P. Conn, Gilles D. Tamagnan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 332 KB

english, 2011

33

Synthesis of a new precursor to the nicotinic receptor tracer 5-IA-85380 precursor using trimethylsilyl iodide as deblocking agent

Eric Brenner, Ronald M Baldwin, Gilles Tamagnan

Journal:

Tetrahedron Letters

Year:

2004

Language:

english

File:

PDF, 262 KB

english, 2004

34

Total synthesis of the marine cytotoxic caulibugulones A–D

David Alagille, Ronald M Baldwin, Gilles D Tamagnan

Journal:

Tetrahedron Letters

Year:

2004

Language:

english

File:

PDF, 245 KB

english, 2004

35

One-step synthesis of 2-arylbenzothiazole (‘BTA’) and -benzoxazole precursors for in vivo imaging of β-amyloid plaques

David Alagille, Ronald M. Baldwin, Gilles D. Tamagnan

Journal:

Tetrahedron Letters

Year:

2005

Language:

english

File:

PDF, 98 KB

english, 2005

36

Cyclopentadienyltricarbonylrheniumbenzazepines: synthesis and binding affinity

Gilles Tamagnan, Ronald M Baldwin, Nora S Kula, Ross J Baldessarini, Robert B Innis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 122 KB

english, 2000

37

Synthesis and monoamine transporter affinity of 2β-carbomethoxy-3β-(2″-, 3″- or 4″-substituted) biphenyltropanes

Gilles Tamagnan, Ronald M Baldwin, Nora S Kula, Ross J Baldessarini, Robert B Innis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 139 KB

english, 2000

38

N-Phthalimidoalkyl derivatives of 2β-carbomethoxy-3β-(4′-iodophenyl)tropane (β-CIT): Brain monoamine transporter affinity

Gilles Tamagnan, John L. Neumeyer, Yigong Gao, Shaoyin Wang, Nora S. Kula, Ross J. Baldessarini

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 226 KB

english, 1997

39

Influence of acetylcholine levels on the binding of a SPECT nicotinic acetylcholine receptor ligand [123I]5-I-A-85380

Masahiro Fujita, Mohammed S. Al-Tikriti, Gilles Tamagnan, Sami S. Zoghbi, Ali Bozkurt, Ronald M. Baldwin, Robert B. Innis

Journal:

Year:

2003

Language:

english

File:

PDF, 86 KB

english, 2003

40

Sex differences in [123I]β-CIT SPECT measures of dopamine and serotonin transporter availability in healthy smokers and nonsmokers

Julie K. Staley, Suchitra Krishnan-Sarin, Sami Zoghbi, Gilles Tamagnan, Masahiro Fujita, John P. Seibyl, Paul K. Maciejewski, Stephanie O'Malley, Robert B. Innis

Journal:

Year:

2001

Language:

english

File:

PDF, 358 KB

english, 2001

41

Decreased Beta2*-nicotinic acetylcholine receptor availability after chronic ethanol exposure in nonhuman primates

Kelly P. Cosgrove, Tracy Kloczynski, Frederic Bois, Brian Pittman, Gilles Tamagnan, John P. Seibyl, John H. Krystal, Julie K. Staley

Journal:

Year:

2010

Language:

english

File:

PDF, 76 KB

english, 2010

42

Whole-body biodistribution, radiation absorbed dose, and brain SPET imaging with [123I]5-I-A-85380 in healthy human subjects

Masahiro Fujita, John P. Seibyl, Bruce D. Vaupel, Gilles Tamagnan, Michele Early, Sami S. Zoghbi, Ronald M. Baldwin, Andrew G. Horti, Andrei O. Koren, Alexey G. Mukhin, Shaukat Khan, Ali Bozkurt, Alan

Journal:

European Journal of Nuclear Medicine and Molecular Imaging

Year:

2002

Language:

english

File:

PDF, 127 KB

english, 2002

43

Quantification of nicotinic acetylcholine receptors in human brain using [123I]5-I-A-85380 SPET

Masahiro Fujita, Masanori Ichise, ChristopherH. Dyck, SamiS. Zoghbi, Gilles Tamagnan, AlexeyG. Mukhin, Ali Bozkurt, Nicholas Seneca, Dnyanesh Tipre, ChristopherC. DeNucci, Hidehiro Iida, D.Bruce Vaupe

Journal:

European Journal of Nuclear Medicine and Molecular Imaging

Year:

2003

Language:

english

File:

PDF, 314 KB

english, 2003

44

[123I]5-IA-85380 SPECT Imaging of β2-Nicotinic Acetylcholine Receptor Availability in the Aging Human Brain

EFFIE M. MITSIS, KELLY P. COSGROVE, JULIE K. STALEY, ERIN B. FROHLICH, FREDERIC BOIS, GILLES D. TAMAGNAN, KRISTINA M. ESTOK, JOHN P. SEIBYL, CHRISTOPHER H. VAN DYCK

Journal:

Annals of the New York Academy of Sciences

Year:

2007

Language:

english

File:

PDF, 49 KB

english, 2007

45

Substituent Effects of N-(1,3-Diphenyl-1H-pyrazol-5-yl)benzamides on Positive Allosteric Modulation of the Metabotropic Glutamate-5 Receptor in Rat Cortical Astrocytes

de Paulis, Tomas, Hemstapat, Kamondanai, Chen, Yelin, Zhang, Yongqin, Saleh, Samir, Alagille, David, Baldwin, Ronald M., Tamagnan, Gilles D., Conn, P. Jeffrey

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 192 KB

english, 2006

46

Iodine-123 labeled reboxetine analogues for imaging of noradrenaline transporter in brain using single photon emission computed tomography

Adriana Alexandre S. Tavares, Nicola K. Jobson, Deborah Dewar, Andrew Sutherland, Sally L. Pimlott, Jeffery Batis, Olivier Barret, John Seibyl, Gilles Tamagnan

Journal:

Year:

2012

Language:

english

File:

PDF, 1.35 MB

english, 2012

47

Biodistribution and dosimetry of123I-mZIENT: a novel ligand for imaging serotonin transporters

Alice Nicol, Rajeev Krishnadas, Sue Champion, Gilles Tamagnan, Jeffrey S. Stehouwer, Mark M. Goodman, Donald M. Hadley, Sally L. Pimlott

Journal:

European Journal of Nuclear Medicine and Molecular Imaging

Year:

2012

Language:

english

File:

PDF, 362 KB

english, 2012

48

Erratum to “Potent mGluR5 antagonists: Pyridyl and thiazolyl-ethynyl-3,5-disubstituted-phenyl series” [Bioorg. Med. Chem. Lett. 21 (2011) 3243–3247]

David Alagille, Herve DaCosta, Yelin Chen, Kamondanai Hemstapat, Alice Rodriguez, Ronald M. Baldwin, P. Jeffrey Conn, Gilles D. Tamagnan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 113 KB

english, 2012

49

Local anesthetic effects of cocaethylene and isopropylcocaine on rat peripheral nerves

Hajime A. Tokuno, Charles W. Bradberry, Brian Everill, Samuel K. Agulian, Steven Wilkes, Ronald M. Baldwin, Gilles D. Tamagnan, Jeffery D. Kocsis

Journal:

Year:

2004

Language:

english

File:

PDF, 236 KB

english, 2004

50

Regional distribution and behavioral correlates of 5-HT2A receptors in Alzheimer's disease with [18F]deuteroaltanserin and PET

Lekshmi Santhosh, Kristina M. Estok, Rebecca S. Vogel, Gilles D. Tamagnan, Ronald M. Baldwin, Effie M. Mitsis, Martha G. MacAvoy, Julie K. Staley, Christopher H. van Dyck

Journal:

Psychiatry Research: Neuroimaging

Year:

2009

Language:

english

File:

PDF, 404 KB

english, 2009

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